| Assay Method Information | |
| | ChEMBL_1735959 (CHEMBL4151495) |
| Description: | Inhibition of N-terminal FLAG-tagged human full-length CDK12 (1 to 1490 residues)/N-terminal His-tagged CycK (1 to 580 residues) expressed in Sf9 cells assessed as reduction in ATP-dependent ULight-4E-BP1 (Thr37/Thr46) substrate peptide phosphorylation pre-incubated for 60 mins by LANCE Ultra assay |
| Affinity data for this assay | |
|---|---|
| If you find an error in this entry please send us an E-mail | |