| Assay Method Information | |
| | ChEMBL_1780729 (CHEMBL4252246) |
| Description: | Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated for 10 mins followed by ATP induction measured after 25 mins by fluorescence assay |
| Affinity data for this assay | |
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