Assay Method Information

Assay Name:  ChEMBL_1873767 (CHEMBL4375056)
Description:  Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-induced cAMP production preincubated for 15 mins followed by isoproterenol addition and measured after 30 mins by TR-FRET assay
Affinity data for this assay
 

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