Assay Method Information

Assay Name:  ChEMBL_2132592 (CHEMBL4842107)
Description:  Partial agonist activity at D3 receptor (unknown origin) expressed in HEK293T cells co-expressing GFP2-beta-arrestin2 assessed as beta-arrestin2 recruitment preincubated for 2 mins with coelenterazine followed by compound addition and measured after 2 mins by BRET assay
Affinity data for this assay
 

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