Assay Method Information

Assay Name:  ChEMBL_1718141 (CHEMBL4133141)
Description:  Antagonist activity at rat P2X7 receptor expressed in human 1321N1 cells assessed as reduction in agonist-induced intracellular Ca2+ levels preincubated for 3 mins followed by agonist addition measured up to 2 mins by Fluo-4 dye-based FLIPR assay
Affinity data for this assay
 

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