Assay Method Information | |
| ChEMBL_1660893 (CHEMBL1249492) |
Description: | Inhibition of CYP2B6 in human liver microsomes assessed as enzyme-mediated metabolite formation using bupropion as substrate incubated for 5 mins followed by NADPH addition measured after 30 mins by LC-MS/MS analysis |
Affinity data for this assay | |
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