Assay Method Information

Assay Name:  ChEMBL_1728754 (CHEMBL4144032)
Description:  Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinylated acetyl-histone H4 peptide and measured after 1 hr by AlphaScreen assay
Affinity data for this assay
 

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