Assay Method Information

Assay Name:  ChEMBL_1778241 (CHEMBL4235233)
Description:  Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pretreated for 5 mins followed by GSK1016790A addition by Fluo-4-AM dye based fluorescence assay
Affinity data for this assay
 

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