| Assay Method Information | |
| | ChEMBL_1656138 (CHEMBL4005608) |
| Description: | Inhibition of recombinant G9a catalytic SET domain (913 to 1193 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) codon plus RIL assessed as inhibition of methylation activity using biotin-labeled H3 (1 to 25 residues) as substrate and [3H]-SAM after 2 hrs by scintillation proximity assay |
| Affinity data for this assay | |
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