Assay Method Information

Assay Name:  ChEMBL_2099984 (CHEMBL4808380)
Description:  Binding affinity to Galphaq/11 (unknown origin) expressed in HEK293 cells cotransfected with AT1R/Galphaq-RLuc8/ Ggamma2-venus/Gbeta1 assessed as inhibition of Ang-II induced-BRET signal preincubated for 1 hr followed by Ang-II addition by BRET assay
Affinity data for this assay
 

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