Assay Method Information | |
| ChEMBL_1660935 (CHEMBL4010547) |
Description: | Inhibition of CYP3A4 in human liver microsomes assessed as enzyme-mediated metabolite formation using testosterone as substrate incubated for 5 mins followed by NADPH addition measured after 30 mins by LC-MS/MS analysis |
Affinity data for this assay | |
---|---|
If you find an error in this entry please send us an E-mail |