| Assay Method Information | |
| | ChEMBL_2046328 (CHEMBL4701027) |
| Description: | Antagonist activity at human adenosine 2A receptor expressed in HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins followed by 5 nM A2A agonist NECA addition and measured after 30 mins by EU-cAMP tracer based TR-FRET assay |
| Affinity data for this assay | |
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