Assay Method Information

Assay Name:  ChEMBL_2033576 (CHEMBL4687734)
Description:  Competitive inhibition of human recombinant CYP3A4 expressed in baculovirus-infected insect cells using diltiazem as substrate incubated for 15 mins followed by NADPH-generating system addition by Michaelis-Menten plot analysis
Affinity data for this assay
 

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