| Assay Method Information | |
| | ChEMBL_1699995 (CHEMBL4050977) |
| Description: | Antagonist activity at human KOR expressed in HEK293T cells coexpressing Gi assessed as Gi-mediated inhibition of cAMP production incubated for 15 mins followed by Gs activator isoproterenol addition measured after 15 mins by luciferase reporter gene assay |
| Affinity data for this assay | |
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