Assay Method Information | |
| ChEMBL_2151352 (CHEMBL758949) |
Description: | Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for 30 mins followed by [3H]-pitavastatin addition and measured after 2 mins by liquid scintillation analysis |
Affinity data for this assay | |
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