Assay Method Information | |
| ChEMBL_1569236 (CHEMBL3791660) |
Description: | Antagonist activity at rat TRPA1 expressed in tetracycline-inducible T-REx expression system transfected CHO cells assessed as inhibition of methylglyoxal-induced 45Ca2+ uptake preincubated for 10 mins followed by methylglyoxal addition measured after 3 mins by TopCount microplate scintillator counting method |
Affinity data for this assay | |
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