| Assay Method Information | |
| | ChEMBL_1661604 (CHEMBL4011216) |
| Description: | Antagonist activity at human dopamine D2 receptor expressed in HEK293 cells assessed as reduction in quinpirole-mediated cAMP inhibition preincubated for 15 mins followed by quinpirole addition measured for 1 sec by BRET assay |
| Affinity data for this assay | |
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