Assay Method Information

Assay Name:  ChEMBL_1660907 (CHEMBL4010519)
Description:  Inhibition of CYP2C9 in human liver microsomes assessed as enzyme-mediated metabolite formation using diclofenac as substrate incubated for 5 mins followed by NADPH addition measured after 30 mins by LC-MS/MS analysis
Affinity data for this assay
 

If you find an error in this entry please send us an E-mail