| Assay Method Information | |
| | ChEMBL_1660880 (CHEMBL4010492) |
| Description: | Inhibition of CYP1A2 in human liver microsomes assessed as enzyme-mediated metabolite formation using phenacetin as substrate incubated for 5 mins followed by NADPH addition measured after 30 mins by LC-MS/MS analysis |
| Affinity data for this assay | |
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