Assay Method Information

Assay Name:  ChEMBL_2669541
Description:  Antagonist activity at eYFP-tagged human GPR1 transfected in HEK293 cells assessed as inhibition of TAMRA-labeled-(RG4)-C9 induced receptor internalization by measuring chemerin 9 EC50 at 30 uM incubated for 1 hrs by high content imaging analysis (Rvb = 4 nM)
Affinity data for this assay
 

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