Assay Method Information

Assay Name:  ChEMBL_1493640 (CHEMBL3530056)
Description:  Metabolism-dependent inhibition of CYP3A4 in human liver microsomes using atorvastatin as substrate preincubated for 20 mins with NADPH prior to initiation of reaction with probe substrate by HPLC analysis
Affinity data for this assay
 

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