| Assay Method Information | |
| | ChEMBL_1661608 (CHEMBL4011220) |
| Description: | Antagonist activity at renilla luciferase-tagged human dopamine D2 receptor expressed in HEK293 cells coexpressing mVenus-fused beta-arrestin 2 assessed as reduction in quinpirole-mediated beta-arrestin 2 recruitment preincubated for 15 mins followed by quinpirole addition measured for 1 sec by BRET assay |
| Affinity data for this assay | |
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