Assay Method Information

Assay Name:  ChEMBL_2161635 (CHEMBL5046496)
Description:  Antagonist activity at human mu opioid receptor expressed in HEK293T cells assessed as Galphai2 activation preincubated with compound in D-PBS for 3 hrs followed by coelenterazine addition for 5 mins once again compound addition for 10 mins by BRET assay
Affinity data for this assay
 

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