Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 1GJA
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14155(N-(4-CARBAMIMIDOYL-PHENYL)-2-HYDROXY-BENZAMIDE | N...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14155(N-(4-CARBAMIMIDOYL-PHENYL)-2-HYDROXY-BENZAMIDE | N...)
Affinity DataKi:  3.80E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)