Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 1LI2
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM26187(CHEMBL14060 | phenol | US9688816, 2 | α-CA in...)
Affinity DataKd:  1.09E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102E double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM26187(CHEMBL14060 | phenol | US9688816, 2 | α-CA in...)
Affinity DataKd:  1.03E+5nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102H double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin(Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM26187(CHEMBL14060 | phenol | US9688816, 2 | α-CA in...)
Affinity DataKd:  9.10E+4nMAssay Description:Binding affinity to Enterobacteria phage T4 lysozyme L99A/M102Q double mutant expressed in Escherichia coli BL21(DE3) by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndolysin [L99A,M102Q](Enterobacteria phage T4)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM26187(CHEMBL14060 | phenol | US9688816, 2 | α-CA in...)
Affinity DataKd:  9.09E+4nMAssay Description:Dissociation constant against T4 lysozyme mutant L99AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)