Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 1UK1
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM27714(CHEMBL361054 | 5-fluoro-1-[4-(4-phenyl-1,2,3,6-tet...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM27714(CHEMBL361054 | 5-fluoro-1-[4-(4-phenyl-1,2,3,6-tet...)
Affinity DataIC50: 60nMpH: 8.0 T: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)