Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) for PDB: 2CHZ
LigandPNGBDBM50042924(CHEMBL1229535)
Affinity DataEC50:  4nMAssay Description:Inhibition of PI3K gamma (unknown origin) by membrane capture assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50042924(CHEMBL1229535)
Affinity DataKi:  7nMAssay Description:Inhibition of PI3K-gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50042924(CHEMBL1229535)
Affinity DataKi:  7nMAssay Description:Binding affinity to PI3Kgamma (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50042924(CHEMBL1229535)
Affinity DataIC50: 16nMAssay Description:Inhibition of PI3Kgamma (unknown origin) using phosphatidylinositol and gamma-32P-ATP incubated for 20 mins by TLC assay or high-throughput membrane ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50042924(CHEMBL1229535)
Affinity DataIC50: 16nMAssay Description:Inhibition of human PI3KCgamma by non-radiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50042924(CHEMBL1229535)
Affinity DataIC50: 17nMAssay Description:Inhibition of histidine-tagged recombinant human full length PI3Kgamma expressed in insect cells preincubated for 15 mins followed by addition of col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)