Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 2O65
TargetSerine/threonine-protein kinase pim-1(Human)
Loma Linda University School of Medicine

Curated by ChEMBL
LigandPNGBDBM26656(5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chrome...)
Affinity DataIC50: 646nMAssay Description:Inhibition of PIM1 kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase pim-1(Human)
Loma Linda University School of Medicine

Curated by ChEMBL
LigandPNGBDBM26656(5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chrome...)
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) expressed in Escherichia coli after 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase pim-1(Human)
Loma Linda University School of Medicine

Curated by ChEMBL
LigandPNGBDBM26656(5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chrome...)
Affinity DataIC50: 650nMpH: 7.0 T: 2°CAssay Description:The 96-well flat-bottomed plates were coated with recombinant GST-BAD. After the plates were blocked, the reaction buffer containing test compound an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)