Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 2P3T
TargetCoagulation factor X(Human)
Berlex Biosciences

LigandPNGBDBM17135(Thiophene-Anthranilamide, 17m | ZK813039 | 3-chlor...)
Affinity DataKi:  0.00500nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCoagulation factor X(Human)
Berlex Biosciences

LigandPNGBDBM17135(Thiophene-Anthranilamide, 17m | ZK813039 | 3-chlor...)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCoagulation factor X(Rat)
Berlex Biosciences

LigandPNGBDBM17135(Thiophene-Anthranilamide, 17m | ZK813039 | 3-chlor...)
Affinity DataKi:  0.0600nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)