Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 2R7B
LigandPNGBDBM19087(15,16-dimethoxy-6-methyl-8,12-diazatetracyclo[8.8....)
Affinity DataIC50: 60nMpH: 7.4 T: 2°CAssay Description:A homogeneous in vitro assay based on a LANCE format was first used for high-throughput screening. Those compounds that showed the largest different...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM19087(15,16-dimethoxy-6-methyl-8,12-diazatetracyclo[8.8....)
Affinity DataIC50: 60nMAssay Description:Inhibition of human GST-tagged-PDK1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM19087(15,16-dimethoxy-6-methyl-8,12-diazatetracyclo[8.8....)
Affinity DataIC50: 60nMAssay Description:Inhibition of PDK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)