Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 2VTJ
LigandPNGBDBM24631(4-[(6-chloropyrazin-2-yl)amino]benzene-1-sulfonami...)
Affinity DataIC50: 1.90E+3nMpH: 7.2 T: 2°CAssay Description:CDK2/cyclin A activity was determined using a radiometric assay to measure the incorporation of gamma-phosphate from [gamma-33P]-ATP into histone H1....More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 2(Human)
Astex Therapeutics

Curated by ChEMBL
LigandPNGBDBM24631(4-[(6-chloropyrazin-2-yl)amino]benzene-1-sulfonami...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)