Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 3TIY
TargetCyclin-dependent kinase 2(Human)
Moffitt Cancer Center

LigandPNGBDBM50088360(Purpurogallin | purpurogalline | 2,3,4,6-tetrahydr...)
Affinity DataIC50: 1.70E+4nMAssay Description:The inhibitory against activated CDK2-cyclin A2 complex was determined by using the ADP Quest fluorescence assay from (DiscoveRX, Fremont, CA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50088360(Purpurogallin | purpurogalline | 2,3,4,6-tetrahydr...)
Affinity DataIC50: 1.70E+4nMAssay Description:Competitive inhibition of human CDK2/cyclinA using PKTPKKAKKL as substrate in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)