Report error Found 4 Enz. Inhib. hit(s) for PDB: 3TUH
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
Fujian Medical University (Fmu)
Curated by ChEMBL
Fujian Medical University (Fmu)
Curated by ChEMBL
Affinity DataKd: 24nMAssay Description:Binding affinity to HSP90 (unknown origin) by fluorescence quenching methodMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
Fujian Medical University (Fmu)
Curated by ChEMBL
Fujian Medical University (Fmu)
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of Hsp90 in human MG63 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
Fujian Medical University (Fmu)
Curated by ChEMBL
Fujian Medical University (Fmu)
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of Hsp90 in human MG63 cellsMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
Fujian Medical University (Fmu)
Curated by ChEMBL
Fujian Medical University (Fmu)
Curated by ChEMBL
Affinity DataIC50: 5.39E+3nMAssay Description:Inhibition of human HSP90More data for this Ligand-Target Pair

3D Structure (crystal)