Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4AL4
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86130(LDHA Inhibitor, 26)
Affinity DataKd:  130nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86130(LDHA Inhibitor, 26)
Affinity DataIC50: 4.20E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)