Report error Found 1 Enz. Inhib. hit(s) for PDB: 4ARK
TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Bayer Healthcare
Curated by ChEMBL
Bayer Healthcare
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of MEK1 (unknown origin) after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair

3D Structure (crystal)