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Report error Found 1 Enz. Inhib. hit(s) for PDB: 4B99
TargetMitogen-activated protein kinase 7(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM199090(XMD17-109 | US9676792, Compound 26)
Affinity DataIC50: 162nM EC50:  90nMpH: 7.5Assay Description:Kinase activity was determined in an assay volume of 40 μl in kinase buffer (50 mM Tris-HCl, pH 7.5, 0.1 mM EGTA, 1 mM 2-mercaptoethanol) contai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
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PDB3D3D Structure (crystal)