Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 4BTM
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandPNGBDBM50506661(CHEMBL4517951)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandPNGBDBM50506661(CHEMBL4517951)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to CM5 sensor chip immobilized C-terminal His6/TEV fused-GST-tagged human TTBK1 (14 to 313 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Csic

Curated by ChEMBL
LigandPNGBDBM50506661(CHEMBL4517951)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to phosphorylated TTBK1 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)