Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4BZ9
TargetHistone deacetylase 8(Blood fluke)
Dipartimento Di Chimica E Tecnologie Del Farmaco "Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50239016(DNDI1416947 | CHEMBL2094337)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of Schistosoma mansoni HDAC8 using Fluor de Lys(R) as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 8(Blood fluke)
Dipartimento Di Chimica E Tecnologie Del Farmaco "Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50239016(DNDI1416947 | CHEMBL2094337)
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of Schistosoma mansoni KDAC8 using (FAM)-labeled peptide as substrate after 60 mins by microfluidic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)