Report error Found 2 Enz. Inhib. hit(s) for PDB: 4EK9
TargetHistone-lysine N-methyltransferase, H3 lysine-79 specific(Human)
Boston University
Curated by ChEMBL
Boston University
Curated by ChEMBL
Affinity DataKi: 9.00E+3nMAssay Description:Inhibition of DOT1-like Histone H3 Methyltransferase (unknown origin)More data for this Ligand-Target Pair
3D Structure (crystal)TargetHistone-lysine N-methyltransferase, H3 lysine-79 specific(Human)
Boston University
Curated by ChEMBL
Boston University
Curated by ChEMBL
Affinity DataKi: 3.80E+4nMAssay Description:Competitive inhibition of recombinant human DOT1L using adenosine/deazaadenosine as substrate and SAM cofactorMore data for this Ligand-Target Pair