Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4F7V
Target2-amino-4-hydroxy-6-hydroxymethyldihydropteridine pyrophosphokinase(Escherichia coli (strain K12))
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50485340(CHEMBL2046607)
Affinity DataKd:  4.16E+3nMAssay Description:Binding affinity to Escherichia coli HPPK at pH 8.3 by fluorometric titrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target2-amino-4-hydroxy-6-hydroxymethyldihydropteridine pyrophosphokinase(Escherichia coli (strain K12))
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50485340(CHEMBL2046607)
Affinity DataIC50: 9.53E+3nMAssay Description:Inhibition of Escherichia coli HPPK using [alpha-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)