Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) for PDB: 4G17
TargetCasein kinase I isoform gamma-2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50390498(CHEMBL2071612)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of CK1gamma2 expressed in HEK293 cells assessed as inhibition of LRP6 Thr1479 phosphorylation by immunoblottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)