Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 4GQ3
TargetMenin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM152235(US8993552, 70)
Affinity DataKd:  158nMAssay Description:Binding affinity to menin (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM152235(US8993552, 70)
Affinity DataIC50: 430nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetMenin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM152235(US8993552, 70)
Affinity DataIC50: 446nMAssay Description:Displacement of FITC-MBM1 from menin (unknown origin) measured after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)