Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4GQ4
TargetMenin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50117750(CHEMBL3586090)
Affinity DataIC50: 46nMAssay Description:Inhibition of N-terminal thioredoxin His6-tagged full-length human menin expressed in Escherichia coli Rosetta (DE3) cells assessed as reduction in m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50117750(CHEMBL3586090)
Affinity DataIC50: 190nMAssay Description:Inhibition of FITC-labelled MLL1 binding to menin (unknown origin) after 120 mins by fluorescence polarization methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)