Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4GVM
TargetIntegrase(Human immunodeficiency virus type 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50011006(CHEMBL3259895)
Affinity DataKd:  150nMAssay Description:Binding affinity to HIV1 integrase by displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetIntegrase(Human immunodeficiency virus type 1)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50011006(CHEMBL3259895)
Affinity DataIC50: 60nMAssay Description:Binding affinity to recombinant HIV-1 integrase catalytic core domain expressed in Escherichia coli assessed as inhibition of interaction with LEDFG/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)