Report error Found 3 Enz. Inhib. hit(s) for PDB: 4HYH
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant His-tagged CHK1 (unknown origin) expressed in baculovirus expression system using biotin-RSGLYRSPSMPENLNRPR as substrate af...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 3.70nMAssay Description:Inhibition of human CHK1More data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of CHK1 in human U2OS cells assessed as phosphorylation of H2AX after 2 hrs by FITC/propidium iodide staining-based immunofluorescence ass...More data for this Ligand-Target Pair