Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4KW5
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50574428(CHEMBL3262462)
Affinity DataIC50: 53nMAssay Description:Inhibition of Mycobacterium tuberculosis wild type DprE1 expressed in Escherichia coli BL21 DE3 assessed as formation of resorufin using FPR as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Northwest A&F University

Curated by ChEMBL
LigandPNGBDBM50574428(CHEMBL3262462)
Affinity DataIC50: 266nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)