Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4MGD
TargetEstrogen receptor(Human)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50410509(SJ000143975 | CHEMBL196585)
Affinity DataEC50:  31nMAssay Description:Agonist activity at ERalpha (unknown origin) expressed in human HeLa cells assessed as transcriptional activation measured after 24 hrs by luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor(Human)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50410509(SJ000143975 | CHEMBL196585)
Affinity DataIC50: 43nMAssay Description:Displacement of [3H]17-beta estradiol from GST-fused human recombinant ERalpha ligand binding domain expressed in Escherichia coli BL21alpha cells in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)