Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4R1Y
TargetHepatocyte growth factor receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50065456(CHEMBL3402741)
Affinity DataIC50: 400nMAssay Description:Inhibition of GST-His6-tagged recombinant human c-Met kinase domain (956 to 1390) after 60 mins by anoff-chip mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50065456(CHEMBL3402741)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of c-Met kinase in human A549 cells assessed as inhibition of phosphorylation after 45 mins by electrochemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)