Report error Found 2 Enz. Inhib. hit(s) for PDB: 4TV3
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
University of Calabria
Curated by ChEMBL
University of Calabria
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of human P13Kalpha assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
University of Calabria
Curated by ChEMBL
University of Calabria
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of human PI3Kalpha assessed as inhibition constantMore data for this Ligand-Target Pair

3D Structure (crystal)