Report error Found 2 Enz. Inhib. hit(s) for PDB: 4XX9
Target3-phosphoinositide-dependent protein kinase 1(Human)
Bioinformatics Institute (Bii)
Curated by ChEMBL
Bioinformatics Institute (Bii)
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of human PDK1 catalytic activity using PIFtide as substrate after 1 hr by phosphor imager analysis in presence of [gamma-32P]-ATP relative...More data for this Ligand-Target Pair
3D Structure (crystal)Target3-phosphoinositide-dependent protein kinase 1(Human)
Bioinformatics Institute (Bii)
Curated by ChEMBL
Bioinformatics Institute (Bii)
Curated by ChEMBL
Affinity DataKd: 8.00E+3nMAssay Description:Displacement of PIFtide from human PDK1 PIF pocket after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair